Non-peptidic,low-internalizingδ-selectiveopioidreceptoragonist;derivativeofSNC80(Cat.No.0764).Doesnottriggeracutedesensitizationoftheanalgesicresponse;reducesCFA-inducedhyperalgesia.Brainpenetrantfollowingsystemicadministration.
M.Wt | 384.94 |
Formula | C23H28N2O.HCl |
Storage | Storeat-20°C |
Purity | ≥97%(HPLC) |
CASNumber | 209808-47-9 |
PubChemID | 76848958 |
InChIKey | OTXTZCLQEGSAMW-UHFFFAOYSA-N |
Smiles | O=C(N(CC)CC)C1=CC=C(/C(C3=CC=CC=C3)=C2CCNCC2)C=C1.Cl |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
Solvent | MaxConc.mg/mL | MaxConc.mM | |
---|---|---|---|
Solubility | |||
DMSO | 38.49 | 100 | |
water | 38.49 | 100 |
Thefollowingdataisbasedontheproductmolecularweight384.94.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
---|---|---|---|
1mM | 2.6mL | 12.99mL | 25.98mL |
5mM | 0.52mL | 2.6mL | 5.2mL |
10mM | 0.26mL | 1.3mL | 2.6mL |
50mM | 0.05mL | 0.26mL | 0.52mL |