Aspecificblockerofthetimedependentdelayedrectifierpotassiumcurrent,devoidofanyβ-adrenoceptorblockingactivity.Exhibitsproarrhythmicandprohypertensiveactivityinvivo.
AM92016hydrochlorideisalsoofferedaspartoftheTocriscreenPlus.FindoutmoreaboutcompoundlibrariesavailablefromTocris.
| M.Wt | 483.84 |
| Formula | C19H24Cl2N2O4S.HCl |
| Storage | DesiccateatRT |
| Purity | ≥98%(HPLC) |
| CASNumber | 133229-11-5 |
| PubChemID | 45073415 |
| InChIKey | TXOARFPCQOBODS-UHFFFAOYSA-N |
| Smiles | Cl.CN(CCC1=CC(Cl)=C(Cl)C=C1)CC(O)COC1=CC=C(NS(C)(=O)=O)C=C1 |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
| Solvent | MaxConc.mg/mL | MaxConc.mM | |
|---|---|---|---|
| Solubility | |||
| DMSO | 48.38 | 100 | |
| ethanol | 48.38 | 100 | |
| water | 24.19 | 50 |
Thefollowingdataisbasedontheproductmolecularweight483.84.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 2.07mL | 10.33mL | 20.67mL |
| 5mM | 0.41mL | 2.07mL | 4.13mL |
| 10mM | 0.21mL | 1.03mL | 2.07mL |
| 50mM | 0.04mL | 0.21mL | 0.41mL |



