Sulphydryl-reactivecompoundthatinhibitsagoNISTandantagonistbindingtoG-protein-coupledreceptors.InhibitsavarietyofGPCRsincludingadenosine,opioid,muscarinic,adrenergicanddopaminergicreceptors(IC50valuesare0.1-1.8μM).
SCH202676hydrobromideisalsoofferedaspartoftheTocriscreenPlus.FindoutmoreaboutcompoundlibrariesavailablefromTocris.
M.Wt | 348.26 |
Formula | C15H13N3S.HBr |
Storage | Desiccateat+4°C |
Purity | ≥99%(HPLC) |
CASNumber | 265980-25-4 |
PubChemID | 9884675 |
InChIKey | YJYGOWVFDGULLL-UHFFFAOYSA-N |
Smiles | CN=C1SN(C3=CC=CC=C3)C(C2=CC=CC=C2)=N/1.Br |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
Solvent | MaxConc.mg/mL | MaxConc.mM | |
---|---|---|---|
Solubility | |||
DMSO | 8.71 | 25mMwithgentlewarming |
Thefollowingdataisbasedontheproductmolecularweight348.26.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
---|---|---|---|
1mM | 2.87mL | 14.36mL | 28.71mL |
5mM | 0.57mL | 2.87mL | 5.74mL |
10mM | 0.29mL | 1.44mL | 2.87mL |
50mM | 0.06mL | 0.29mL | 0.57mL |