InhibitsGsandstimulatesGiactivity.InhibitsproteinkinaseCandcAMP-dependentproteinkinases.Na+/K+ATPaseinhibitor.
| M.Wt | 2847 |
| Formula | C131H229N39O31 |
| Sequence | GIGAVLKVLTTGLPALISWIKRKRQQ (Modifications:Gln-26=C-terminalamide) |
| Storage | Desiccateat-20°C |
| CASNumber | 20449-79-0 |
| PubChemID | 16133648 |
| InChIKey | VDXZNPDIRNWWCW-JFTDCZMZSA-N |
| Smiles | [H]NCC(=O)N[C@@H]([C@@H](C)CC)C(=O)NCC(=O)N[C@@H](C)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H]([C@@H](C)O)C(=O)NCC(=O)N[C@@H](CC(C)C)C(=O)N1CCC[C@H]1C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC1=CNC2=C1C=CC=C2)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCC(N)=O)C(N)=O |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
| Solubility | Solubleto1mg/mlinwater |
Thefollowingdataisbasedontheproductmolecularweight2847.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 0.35mL | 1.76mL | 3.51mL |
| 5mM | 0.07mL | 0.35mL | 0.7mL |
| 10mM | 0.04mL | 0.18mL | 0.35mL |
| 50mM | 0.01mL | 0.04mL | 0.07mL |



