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主营:分子类,蛋白类,抗体类,生化类试剂
℡ 4000-520-616
℡ 4000-520-616
Tocris/3-MPPI/0581/50/50 mg
产品编号:0581/50
市  场 价:¥12900.00
场      地:美国(厂家直采)
产品分类: 生化试剂>生物分子>受体>
联系QQ:1570468124
电话号码:4000-520-616
邮      箱: info@ebiomall.com
美  元  价:$645.00
品      牌: Tocris
公      司:Tocris Bioscience
公司分类:
Tocris/3-MPPI/0581/50/50 mg
商品介绍
Description:α1ligand
ChemicalName:2-[(4-Phenylpiperazin-1-yl)methyl]-2,3-dihydroimidazo[1,2-c]quinazolin-5(6H)-one
BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

Verypotentligandforα1sites(Kifordisplacementofprazosin=0.2nM).Displaysdifferentbindingpropertiesforeachα1subtype(pKivaluesare8.74,9.44and9.57forα1B,α1Dandα1Aadrenoceptorsrespectively).Alsobindsto5-HT1Asites(Ki=50nM).

TechnicalData

M.Wt419.48
FormulaC23H25N5O3
StorageStoreatRT
CASNumber133399-65-2
PubChemID4013695
InChIKeyAQASGOHUMGAWJJ-UHFFFAOYSA-N
SmilesCOC1=C(C=CC=C1)N1CCN(CCN2C(=O)NC3=C(NC4=CC=CC=C34)C2=O)CC1

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

SolventMaxConc.mg/mLMaxConc.mM
Solubility
DMSO4.1910mMwithgentlewarming

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight419.48.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass1mg5mg10mg
1mM2.38mL11.92mL23.84mL
5mM0.48mL2.38mL4.77mL
10mM0.24mL1.19mL2.38mL
50mM0.05mL0.24mL0.48mL

ProductDatasheets

CertificateofAnalysisiscurrentlyunavailable
on-line.PleasecontactCustomerService
SafetyDatasheet