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主营:分子类,蛋白类,抗体类,生化类试剂
℡ 4000-520-616
℡ 4000-520-616
Tocris/GSK 0660/3433/10/10 mg
产品编号:3433/10
市  场 价:¥3780.00
场      地:美国(厂家直采)
产品分类: 生化试剂>生物分子>受体>
联系QQ:1570468124
电话号码:4000-520-616
邮      箱: info@ebiomall.com
美  元  价:$189.00
品      牌: Tocris
公      司:Tocris Bioscience
公司分类:
Tocris/GSK 0660/3433/10/10 mg
商品介绍
Description:SelectivePPARδantagoNIST
ChemicalName:3-[[[2-Methoxy-4-(phenylamino)phenyl]amino]sulfonyl]-2-thiophenecarboxylicacidmethylester
Purity:≥99%(HPLC)
BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

SelectivePPARδantagonist(IC50valuesare0.155,>10and10μMatPPARδ,PPARαandPPARγrespectively).Exhibitsinverseagonisteffectswhenadministeredbyitself.

CompoundLibraries

GSK0660isalsoofferedaspartoftheTocriscreenPlus.FindoutmoreaboutcompoundlibrariesavailablefromTocris.

TechnicalData

M.Wt418.49
FormulaC19H18N2O5S2
StorageStoreat+4°C
Purity≥99%(HPLC)
CASNumber1014691-61-2
PubChemID46233311
InChIKeyNDFKBGWLUHKMFY-UHFFFAOYSA-N
SmilesO=S(NC1=C(OC)C=C(NC3=CC=CC=C3)C=C1)(C2=C(C(OC)=O)SC=C2)=O

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

SolventMaxConc.mg/mLMaxConc.mM
Solubility
DMSO41.85100
ethanol4.1810

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight418.49.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass1mg5mg10mg
1mM2.39mL11.95mL23.9mL
5mM0.48mL2.39mL4.78mL
10mM0.24mL1.19mL2.39mL
50mM0.05mL0.24mL0.48mL

ProductDatasheets

CertificateofAnalysis/ProductDatasheet
SafetyDatasheet