ReversIBLeinhibitorofvesiculartraffickingbetweenendoplasmicreticulumandGolgiapparatus.ModifiesGolgiADP-ribosylationfactor(ARF)1GTPaseactivityandinhibitsexocytosis(IC50~20mM).Hassimilar,butnotidentical,actiontobrefeldinA(Cat.No.1231).
Exo1isalsoofferedaspartoftheTocriscreenPlus.FindoutmoreaboutcompoundlibrariesavailablefromTocris.
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
Thefollowingdataisbasedontheproductmolecularweight273.26.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.