请使用支持JavaScript的浏览器!
主营:分子类,蛋白类,抗体类,生化类试剂
℡ 4000-520-616
℡ 4000-520-616
Tocris/Cinalukast/2025/50/50 mg
产品编号:2025/50
市  场 价:¥14100.00
场      地:美国(厂家直采)
产品分类: 生化试剂>生物分子>受体>
联系QQ:1570468124
电话号码:4000-520-616
邮      箱: info@ebiomall.com
美  元  价:$705.00
品      牌: Tocris
公      司:Tocris Bioscience
公司分类:
Tocris/Cinalukast/2025/50/50 mg
商品介绍
Description:Potent,selectiveCysLT1(LTD4)antagoNIST;orallyactive
AlternativeNames:Ro24-5913
ChemicalName:4-[[3-[(1E)-2-(4-Cyclobutyl-2-thiazolyl)ethenyl]phenyl]amino]-2,2-diethyl-4-oxobutanoicacid
Purity:≥98%(HPLC)
BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

Potent,selectiveCysLT1(LTD4)leukotrienereceptorantagonist(IC50=6.4nM).InhibitsLTD4-inducedbronchoconstrictioninguineapigswhenadministeredintravenously,orallyorbyaerosol.

CompoundLibraries

CinalukastisalsoofferedaspartoftheTocriscreenPlus.FindoutmoreaboutcompoundlibrariesavailablefromTocris.

TechnicalData

M.Wt412.55
FormulaC23H28N2O3S
StorageDesiccateat-20°C
Purity≥98%(HPLC)
CASNumber128312-51-6
PubChemID6436135
InChIKeyBZMKNPGKXJAIDV-VAWYXSNFSA-N
SmilesCCC(CC)(CC(=O)NC1=CC(C=CC2=NC(=CS2)C2CCC2)=CC=C1)C(O)=O

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

SolventMaxConc.mg/mLMaxConc.mM
Solubility
DMSO41.26100
ethanol4.1310

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight412.55.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass1mg5mg10mg
1mM2.42mL12.12mL24.24mL
5mM0.48mL2.42mL4.85mL
10mM0.24mL1.21mL2.42mL
50mM0.05mL0.24mL0.48mL

ProductDatasheets

CertificateofAnalysis/ProductDatasheet
SafetyDatasheet