请使用支持JavaScript的浏览器!
主营:分子类,蛋白类,抗体类,生化类试剂
℡ 4000-520-616
℡ 4000-520-616
Tocris/Capsazepine/0464/10/10 mg
产品编号:0464/10
市  场 价:¥3180.00
场      地:美国(厂家直采)
联系QQ:1570468124
电话号码:4000-520-616
邮      箱: info@ebiomall.com
美  元  价:$159.00
品      牌: Tocris
公      司:Tocris Bioscience
公司分类:
Tocris/Capsazepine/0464/10/10 mg
商品介绍
Description:VanilloidreceptorantagoNIST;alsoactivatorofENaCδ
ChemicalName:N-[2-(4-Chlorophenyl)ethyl]-1,3,4,5-tetrahydro-7,8-dihydroxy-2H-2-benzazepine-2-carbothioamide
Purity:≥99%(HPLC)
BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

Selectivevanilloidreceptorantagonist(Ki=3.2μM).Inhibitscarrageenaninflammation-inducedhyperalgesicresponsesintherat.Alsoactivatesamiloride-sensitiveepithelialNa+channelENaCδ.AlsoavailableaspartoftheVanilloidTRPV1ReceptorTocriset™.

CompoundLibraries

CapsazepineisalsoofferedaspartoftheTocriscreenPlus.FindoutmoreaboutcompoundlibrariesavailablefromTocris.

TechnicalData

M.Wt376.9
FormulaC19H21ClN2O2S
StorageStoreatRT
Purity≥99%(HPLC)
CASNumber138977-28-3
PubChemID2733484
InChIKeyDRCMAZOSEIMCHM-UHFFFAOYSA-N
SmilesOC1=C(O)C=C2CN(CCCC2=C1)C(=S)NCCC1=CC=C(Cl)C=C1

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

SolventMaxConc.mg/mLMaxConc.mM
Solubility
DMSO37.69100
ethanol9.4225

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight376.9.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass1mg5mg10mg
1mM2.65mL13.27mL26.53mL
5mM0.53mL2.65mL5.31mL
10mM0.27mL1.33mL2.65mL
50mM0.05mL0.27mL0.53mL

ProductDatasheets

CertificateofAnalysis/ProductDatasheet
SafetyDatasheet