Aselectiveκ-opioidreceptorantagonist.
SoldwiththepermissionoftheUniversityofMinnesota
nor-BinaltorphiminedihydrochlorideisalsoofferedaspartoftheTocriscreenPlus.FindoutmoreaboutcompoundlibrariesavailablefromTocris.
M.Wt | 734.72 |
Formula | C40H43N3O6.2HCl |
Storage | StoreatRT |
Purity | ≥98%(HPLC) |
CASNumber | 113158-34-2 |
PubChemID | 11957626 |
InChIKey | JOJPJLHRMGPDPV-LZQROVCBSA-N |
Smiles | OC1=CC=C2C([C@]34CCN5CC6CC6)=C1O[C@H]4C%11=C(C7=C(N%11)[C@H]%10[C@@]8(CC%13)[C@@]([C@H](N%13CC%12CC%12)CC9=C8C(O%10)=C(O)C=C9)(O)C7)C[C@@]3(O)[C@H]5C2.Cl.Cl |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
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Solvent | MaxConc.mg/mL | MaxConc.mM | |
---|---|---|---|
Solubility | |||
phosphatebufferedsaline | 36.74 | 50mMwithgentlewarming | |
DMSO | 18.37 | 25 | |
water | 18.37 | 25mMwithgentlewarming |
Thefollowingdataisbasedontheproductmolecularweight734.72.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
---|---|---|---|
1mM | 1.36mL | 6.81mL | 13.61mL |
5mM | 0.27mL | 1.36mL | 2.72mL |
10mM | 0.14mL | 0.68mL | 1.36mL |
50mM | 0.03mL | 0.14mL | 0.27mL |