CannABInoidCB1andvanilloidTRPV1(VR1)agonist(Kivaluesare0.5and0.3μMrespectively).Alsoinhibitstheanandamidetransporter(IC50=3.6μM).Analgesic,vasodilatoryandanti-inflammatoryinvivo.
| M.Wt | 439.64 |
| Formula | C28H41NO3 |
| Storage | Desiccateat-20°C |
| Purity | ≥98%(HPLC) |
| CASNumber | 128007-31-8 |
| PubChemID | 6449767 |
| InChIKey | QVLMCRFQGHWOPM-ZKWNWVNESA-N |
| Smiles | O=C(NCC1=CC=C(O)C(OC)=C1)CCCC=C/CC=C/C/C=CC/C=CCCCCC |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
| Solubility | Solubleinethanol(suppliedpre-dissolvedinanhydrousethanol,5mg/ml) |
Thefollowingdataisbasedontheproductmolecularweight439.64.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 2.27mL | 11.37mL | 22.75mL |
| 5mM | 0.45mL | 2.27mL | 4.55mL |
| 10mM | 0.23mL | 1.14mL | 2.27mL |
| 50mM | 0.05mL | 0.23mL | 0.45mL |



