Potentandselectiveμ-opioidreceptoragonist(Kivaluesare7.0,151and470nMforμ-,δ-andκ-opioidreceptorsrespectively).Displaysantinociceptiveactivityinvivo.
M.Wt | 528.59 |
Formula | C22H28N2O.C6H8O7 |
Storage | StoreatRT |
Purity | ≥99%(HPLC) |
CASNumber | 990-73-8 |
PubChemID | 13810 |
InChIKey | IVLVTNPOHDFFCJ-UHFFFAOYSA-N |
Smiles | O=C(O)C(O)(CC(O)=O)CC(O)=O.O=C(CC)N(C3=CC=CC=C3)C1CCN(CCC2=CC=CC=C2)CC1 |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
Solvent | MaxConc.mg/mL | MaxConc.mM | |
---|---|---|---|
Solubility | |||
water | 21.14 | 40 |
Thefollowingdataisbasedontheproductmolecularweight528.59.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
---|---|---|---|
1mM | 1.89mL | 9.46mL | 18.92mL |
5mM | 0.38mL | 1.89mL | 3.78mL |
10mM | 0.19mL | 0.95mL | 1.89mL |
50mM | 0.04mL | 0.19mL | 0.38mL |
Thereconstitutioncalculatorallowsyoutoquicklycalculatethevolumeofareagenttoreconstituteyourvial.Simplyenterthemassofreagentandthetargetconcentrationandthecalculatorwilldeterminetherest.