Endogenousσ1receptorligandandpsychoactiveplantcompound(Ki=14.8μM).Bindingtoσ1inhibitsvoltage-gatedNa+channelsandisresponsIBLeforthebehavioraleffectsofDMT.Alsoa5-HT2Areceptoragonistandinhibitorof5-HTuptakeatplasmamembraneSEROtonintransporters(SERT)(Ki=4.0μM).
M.Wt | 188.27 |
Formula | C12H16N2 |
Storage | Storeat-20°C |
Purity | ≥99%(HPLC) |
CASNumber | 61-50-7 |
PubChemID | 6089 |
InChIKey | DMULVCHRPCFFGV-UHFFFAOYSA-N |
Smiles | CN(CCC2=CNC1=CC=CC=C12)C |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
Solvent | MaxConc.mg/mL | MaxConc.mM | |
---|---|---|---|
Solubility | |||
ethanol | 0.94 | 5 |
Thefollowingdataisbasedontheproductmolecularweight188.27.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
---|---|---|---|
1mM | 5.31mL | 26.56mL | 53.12mL |
5mM | 1.06mL | 5.31mL | 10.62mL |
10mM | 0.53mL | 2.66mL | 5.31mL |
50mM | 0.11mL | 0.53mL | 1.06mL |
Thereconstitutioncalculatorallowsyoutoquicklycalculatethevolumeofareagenttoreconstituteyourvial.Simplyenterthemassofreagentandthetargetconcentrationandthecalculatorwilldeterminetherest.