Highaffinityadeninereceptoragonist(Ki=18nMatratadeninereceptor).Inhibitsforskolin-stimulatedcAMPformationinCHOcellstransfectedwiththeadeninereceptor;alsostimulatesGTPγSbinding(pEC50valuesare8.54and7.21respectively).
M.Wt | 171.59 |
Formula | C5H5N5.HCl |
Storage | DesiccateatRT |
Purity | ≥99%(HPLC) |
CASNumber | 6055-72-7 |
PubChemID | 76219 |
InChIKey | UQVDQSWZQXDUJB-UHFFFAOYSA-N |
Smiles | NC1=C2C(NC=N2)=NC=N1.Cl |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
Solvent | MaxConc.mg/mL | MaxConc.mM | |
---|---|---|---|
Solubility | |||
DMSO | 17.16 | 100 | |
water | 17.16 | 100 |
Thefollowingdataisbasedontheproductmolecularweight171.59.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
---|---|---|---|
1mM | 5.83mL | 29.14mL | 58.28mL |
5mM | 1.17mL | 5.83mL | 11.66mL |
10mM | 0.58mL | 2.91mL | 5.83mL |
50mM | 0.12mL | 0.58mL | 1.17mL |